Metadol 100mg

Product Description

Metadol 100mg is a powerful prescription medicine primarily used for the management of moderate to severe acute pain. It is used to treat Its active ingredient, Tapentadol, is a centrally acting analgesic that offers dual-action relief it works both as an opioid receptor agonist and a norepinephrine reuptake inhibitor. This dual mechanism makes Metadol 100 mg highly effective in treating pain caused by injuries, surgical procedures, musculoskeletal disorders, and certain neuropathic conditions.

What is Metadol 100mg

Metadol 100mg tablets contain Tapentadol 100 mg, a novel synthetic analgesic classified as an atypical Schedule II opioid medication. Unlike traditional opioids such as morphine, Tapentadol is structurally and pharmacologically unique, yet it provides powerful pain relief with a potentially reduced risk of gastrointestinal and respiratory side effects. As a narcotic pain reliever, Metadol 100 mg works on the central nervous system by blocking pain signals and altering the body’s perception of pain. This dual mechanism of action makes it highly effective in managing moderate to severe acute pain, particularly when other non-opioid painkillers fail to provide adequate relief.

Uses of Metadol 100 mg

Metadol 100mg tablet is prescribed to treat various types of pain, including:

• Moderate to severe acute pain (e.g., post-surgical pain)
• Pain from musculoskeletal injuries
• Chronic pain conditions where opioids are necessary
• Neuropathic pain, such as diabetic peripheral neuropathy
• Postoperative pain
• Lower back pain or joint pain due to arthritis or strain

Tapentadol is especially effective when other non-opioid painkillers (like NSAIDs or acetaminophen) are not providing enough relief.

How Does Tapentadol Work

Tapentadol drug in Metadol 100mg tabs works through two complementary mechanisms:

1. Mu-opioid receptor agonist: It binds to opioid receptors in the brain and spinal cord to block pain signals.

2. Norepinephrine reuptake inhibitor (NRI): It increases norepinephrine levels, enhancing the body’s natural pain-inhibition pathways.

This combination makes it more efficient for certain types of neuropathic pain, where standard opioids may not be sufficient.

Dosage and Administration

• Typical dosage: 100 mg taken every 4 to 6 hours as needed for pain.
• Always follow your doctor’s instructions regarding dosage.
• It can be taken with or without food.
• Do not exceed the recommended daily dose (usually not more than 600 mg/day).

Important: Do not suddenly stop using Metadol tablets without medical advice, as it may cause withdrawal symptoms.

Substitutes and Strengths

• Tapenax ER 100mg
• Tapfree ER 100mg

Warnings and Precautions

Metadol 100 (Tapentadol) should be used with caution in:

• Individuals with a history of substance abuse or opioid addiction
• Patients with severe liver or kidney impairment
• Those taking MAO inhibitors or CNS depressants
• Elderly patients (risk of dizziness and falls)
• People with seizure disorders

Who Should Avoid Metadol

Avoid Metadol 100mg if you:

• Are allergic to Tapentadol
• Have severe respiratory depression
• Suffer from paralytic ileus
• Are taking monoamine oxidase inhibitors (MAOIs)

Always inform your doctor about your full medical history before starting this medication.

Drug Interactions

Metadol (Tapentadol) may interact with:

• Alcohol and sedatives: increases risk of CNS depression
• Antidepressants: risk of serotonin syndrome
• MAOIs: contraindicated
• Antihistamines and antipsychotics: may worsen drowsiness or confusion

Side Effects of Metadol Tablet

Common side effects include:

• Dizziness or lightheadedness
• Nausea and vomiting
• Constipation
• Drowsiness or sedation
• Dry mouth
• Headache

Serious side effects (seek medical help immediately):

• Breathing difficulties
• Seizures
• Hallucinations
• Low blood pressure or fainting
• Symptoms of serotonin syndrome (fever, agitation, tremors)

Storage Instructions of Metadol 100

• Store Metadol 100 at room temperature (15°C–30°C)
• Keep it away from children and pets
• Protect from moisture and direct sunlight

Metadol 100 mg is a highly effective pain reliever for patients who do not respond to non-opioid medications. Thanks to Tapentadol’s dual action, it addresses both nociceptive and neuropathic pain efficiently. However, due to its opioid properties, this medicine must be used with care, under strict medical supervision, and never self-medicated.

Additional information